| 摘要 |
The invention provides a method for radiofluorination of biological vecto rs such as peptides comprising reaction of a compound of formula (II): or a salt thereof with a source of [18F]-fluoride, to give a compound of formula (I): or a salt thereof. The method may be effected under mild reaction condi tions and offers a more chemoselective labelling approach Novel reagents for use in the radiofluoridation method, and uses of the resultant 18F-labelled vectors are also provided
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