发明名称 |
NEW CRYSTAL FORM OF TOPIROXOSTAT, AND PREPARATION METHOD THEREFOR |
摘要 |
The present invention relates to a new crystal form of 5-(2-cyan-4-pyridyl)-3-(4-pyridyl)-1,2,4-triazole, and a preparation method therefor. The new crystal form provided in the present invention can be used for treating gout and hyperuricemia. The new crystal form provided in the present invention has good stability, an obvious refinement effect in process, and has a solubility and hygroscopicity satisfying drug use requirements. The crystal form A provided in the present invention has favorable performance facilitating industrial production, and has important value for further optimization and development of the drug. |
申请公布号 |
WO2016155631(A1) |
申请公布日期 |
2016.10.06 |
申请号 |
WO2016CN77887 |
申请日期 |
2016.03.30 |
申请人 |
CRYSTAL PHARMATECH CO., LTD |
发明人 |
CHEN, Minhua;ZHANG, Yanfeng;LIU, Kai;ZHANG, Xiaoyu |
分类号 |
C07D401/14;A61K31/444;A61P19/06;A61P43/00 |
主分类号 |
C07D401/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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