A method for producing HIV maturation inhibitor compound is set forth using betulin Chemical Structure (I) as starting material, and utilizing Lossen rearrangement techniques.
申请公布号
WO2016168447(A1)
申请公布日期
2016.10.20
申请号
WO2016US27504
申请日期
2016.04.14
申请人
VIIV HEALTHCARE (No.4) LIMITED
发明人
ORTIZ, Adrian;SOUMEILLANT, Maxime;SAVAGE, Scott A.;STROTMAN, Neil A.;EASTGATE, Martin D.;HALEY, Matthew W.;HO, Jeanne;NYE, Jeffrey A.;XU, Zhongmin;KIAU, Susanne;BENKOVICS, Tamas;TAN, Yichen