发明名称 |
NEW INDOLIZINE DERIVATIVES, METHOD FOR PREPARING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM FOR THE TREATMENT OF CANCER |
摘要 |
Compounds of formula (I): wherein Ra, Rb, Rc, Rd, R1, R2, R3, R4, R5, X, Y and Het are as defined in the description. Medicinal products containing the same which are useful in treating pathologies involving a deficit in apoptosis, such as cancer, auto-immune diseases, and diseases of the immune system. |
申请公布号 |
EP2807159(B1) |
申请公布日期 |
2016.11.23 |
申请号 |
EP20130704189 |
申请日期 |
2013.01.23 |
申请人 |
LES LABORATOIRES SERVIER;VERNALIS (R&D) LTD. |
发明人 |
LE DIGUARHER, THIERRY;CASARA, PATRICK;STARCK, JÉRÔME-BENOÎT;HENLIN, JEAN-MICHEL;DAVIDSON, JAMES EDWARD PAUL;MURRAY, JAMES BROOKE;GRAHAM, CHRISTOPHER JOHN;CHEN, I-JEN;GENESTE, OLIVIER;HICKMAN, JOHN;DEPIL, STÉPHANE;LE TIRAN, ARNAUD;NYERGES, MIKLOS;DE NANTEUIL, GUILLAUME |
分类号 |
C07D471/04;A61K31/407;A61K31/4353;A61K31/436;A61P35/00;A61P37/00;C07D487/04;C07D491/052 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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