发明名称 NEW INDOLIZINE DERIVATIVES, METHOD FOR PREPARING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM FOR THE TREATMENT OF CANCER
摘要 Compounds of formula (I): wherein Ra, Rb, Rc, Rd, R1, R2, R3, R4, R5, X, Y and Het are as defined in the description. Medicinal products containing the same which are useful in treating pathologies involving a deficit in apoptosis, such as cancer, auto-immune diseases, and diseases of the immune system.
申请公布号 EP2807159(B1) 申请公布日期 2016.11.23
申请号 EP20130704189 申请日期 2013.01.23
申请人 LES LABORATOIRES SERVIER;VERNALIS (R&D) LTD. 发明人 LE DIGUARHER, THIERRY;CASARA, PATRICK;STARCK, JÉRÔME-BENOÎT;HENLIN, JEAN-MICHEL;DAVIDSON, JAMES EDWARD PAUL;MURRAY, JAMES BROOKE;GRAHAM, CHRISTOPHER JOHN;CHEN, I-JEN;GENESTE, OLIVIER;HICKMAN, JOHN;DEPIL, STÉPHANE;LE TIRAN, ARNAUD;NYERGES, MIKLOS;DE NANTEUIL, GUILLAUME
分类号 C07D471/04;A61K31/407;A61K31/4353;A61K31/436;A61P35/00;A61P37/00;C07D487/04;C07D491/052 主分类号 C07D471/04
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