发明名称 |
PROCESS FOR PREPARING PHARMACEUTICAL COMPOUNDS |
摘要 |
Cryptophycin compounds may be prepared utilizing an epoxidation step early in the synthetic process under the conditions set forth herein. This invention also relates to novel intermediates generated by this early epoxidation process. |
申请公布号 |
CA2281108(A1) |
申请公布日期 |
1998.09.03 |
申请号 |
CA19982281108 |
申请日期 |
1998.02.25 |
申请人 |
UNIVERSITY OF HAWAII;ELI LILLY AND COMPANY;WAYNE STATE UNIVERSITY |
发明人 |
HOARD, DAVID WARREN;MOHER, ERIC DAVID;PATEL, VINOD FRANCIS |
分类号 |
C07D303/16;A61K31/395;A61P35/00;C07C229/08;C07C271/22;C07D233/54;C07D277/30;C07D301/03;C07D303/38;C07D303/40;C07D303/46;C07D405/06;C07D405/12;C07D413/06;C07F7/18 |
主分类号 |
C07D303/16 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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