发明名称 |
METHOD FOR PREPARING THE ANHYDROUS CRYSTALLINE FORM OF ISONIAZID-DERIVED HYDRAZONE, THUS PRODUCED CRYSTALLINE POLYMORPH OF THE ANHYDROUS FORM, USE THEREOF FOR THE TREATMENT OF ALZHEIMER'S DISEASE, PARKINSONISM AND OTHER NEURODEGENERATIVE DISORDERS, AND PHARMACEUTICAL COMPOSITION |
摘要 |
The present invention relates to the method for preparing the anhydrous crystalline form of isoniazid-derived hydrazone (8-hydroxyquinoline-2-carboxaldehyde isonicotinoyl hydrazone), to the thus produced polymorph and to the use thereof for the treatment of Alzheimer's disease and parkinsonism, inter alia, and to a pharmaceutical composition. |
申请公布号 |
EP3085691(A1) |
申请公布日期 |
2016.10.26 |
申请号 |
EP20140872636 |
申请日期 |
2014.06.06 |
申请人 |
FACULDADES CATÓLICAS, ASSOCIAÇÃO SEM FINS LUCRATIVOS, MANTENEDORA DA PONTIFÍCIA UNIVERSIDADE CATÓLICA |
发明人 |
REY, NICOLÁS ADRIÁN;VIANA DE FREITAS, LEONARDO |
分类号 |
C07D215/24;A61K31/4409;A61K31/47;A61P25/00;A61P25/16;A61P25/28;C07D213/86 |
主分类号 |
C07D215/24 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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