摘要 |
<p>A series of 5,6-dihydro-1-benzothiophen-7(4H)-one derivatives, and analogues thereof, which are substituted in the 2-position by an optionally substituted morpholin-4-yl moiety, being selective inhibitors of PI3 kinase enzymes, are accordingly of benefit in medicine, for example in the treatment of inflammatory, autoimmune, cardiovascular, neurodegenerative, metabolic, oncological, nociceptive or ophthalmic conditions.</p> |
申请人 |
UCB PHARMA S.A.;ALEXANDER, RIKKI PETER;BAILEY, STUART;BRAND, STEPHEN;BROOKINGS, DANIEL CHRISTOPHER;BROWN, JULIEN ALISTAIR;HAUGHAN, ALAN FINDLAY;KINSELLA, NATASHA;LOWE, CHRISTOPHER;MACK, STEPHEN ROBERT;PITT, WILLIAM ROSS;RICHARD, MARIANNA DILANI;SHARPE, ANDREW;TAIT, LAURA JANE |
发明人 |
ALEXANDER, RIKKI PETER;BAILEY, STUART;BRAND, STEPHEN;BROOKINGS, DANIEL CHRISTOPHER;BROWN, JULIEN ALISTAIR;HAUGHAN, ALAN FINDLAY;KINSELLA, NATASHA;LOWE, CHRISTOPHER;MACK, STEPHEN ROBERT;PITT, WILLIAM ROSS;RICHARD, MARIANNA DILANI;SHARPE, ANDREW;TAIT, LAURA JANE |