发明名称 FUSED THIOPHENE DERIVATIVES AS KINASE INHIBITORS
摘要 <p>A series of 5,6-dihydro-1-benzothiophen-7(4H)-one derivatives, and analogues thereof, which are substituted in the 2-position by an optionally substituted morpholin-4-yl moiety, being selective inhibitors of PI3 kinase enzymes, are accordingly of benefit in medicine, for example in the treatment of inflammatory, autoimmune, cardiovascular, neurodegenerative, metabolic, oncological, nociceptive or ophthalmic conditions.</p>
申请公布号 WO2007141504(A1) 申请公布日期 2007.12.13
申请号 WO2007GB02051 申请日期 2007.06.04
申请人 UCB PHARMA S.A.;ALEXANDER, RIKKI PETER;BAILEY, STUART;BRAND, STEPHEN;BROOKINGS, DANIEL CHRISTOPHER;BROWN, JULIEN ALISTAIR;HAUGHAN, ALAN FINDLAY;KINSELLA, NATASHA;LOWE, CHRISTOPHER;MACK, STEPHEN ROBERT;PITT, WILLIAM ROSS;RICHARD, MARIANNA DILANI;SHARPE, ANDREW;TAIT, LAURA JANE 发明人 ALEXANDER, RIKKI PETER;BAILEY, STUART;BRAND, STEPHEN;BROOKINGS, DANIEL CHRISTOPHER;BROWN, JULIEN ALISTAIR;HAUGHAN, ALAN FINDLAY;KINSELLA, NATASHA;LOWE, CHRISTOPHER;MACK, STEPHEN ROBERT;PITT, WILLIAM ROSS;RICHARD, MARIANNA DILANI;SHARPE, ANDREW;TAIT, LAURA JANE
分类号 C07D333/66;A61K31/5377;A61K31/55;A61P3/00;C07D333/68;C07D409/12;C07D409/14;C07D451/04;C07D453/02;C07D471/04;C07D495/04 主分类号 C07D333/66
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