发明名称 |
Substituted Quinazoline or Pyridopyrimidine Derivative |
摘要 |
The present invention provides a compound having a glucokinase activating action being useful for prevention or treatment of diabetes mellitus, etc. being represented by the formula (I): X is nitrogen atom, etc.; Y is oxygen atom, etc.; R<SUP>1 </SUP>is an optionally substituted five to six-membered heteroaryl group, etc.; R<SUP>2 </SUP>is hydrogen atom or fluorine atom; and ring A is a monocyclic or bicyclic heteroaryl group which may have a substituent represented by the formula (II)] or a pharmaceutically acceptable salt thereof.
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申请公布号 |
US2008032996(A1) |
申请公布日期 |
2008.02.07 |
申请号 |
US20050593540 |
申请日期 |
2005.03.23 |
申请人 |
MITSUYA MORIHIRO;BAMBA MAKOTO;SASAKI YASUHIRO;NISHIMURA TERUYUKI;EIKI JUN-ICHI;ARAKAWA KEISUKE |
发明人 |
MITSUYA MORIHIRO;BAMBA MAKOTO;SASAKI YASUHIRO;NISHIMURA TERUYUKI;EIKI JUN-ICHI;ARAKAWA KEISUKE |
分类号 |
A61K31/519;A61K31/513;A61K31/517;A61K38/28;A61K45/00;A61P3/04;A61P3/10;A61P9/10;A61P13/12;A61P25/28;A61P27/02;A61P43/00;C07D401/14;C07D403/12;C07D403/14;C07D405/14;C07D413/12;C07D413/14;C07D417/14;C07D471/04;C07D513/04;C07D519/00 |
主分类号 |
A61K31/519 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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