发明名称 Substituted azines as pesticides
摘要 The invention relates to compounds of the general formula (I), wherein the variable have the meanings as indicated in the claims, or a physiologically acceptable salt thereof. The active ingredients have advantageous pesticidal properties. They are especially suitable for controlling endoparasites in warm-blooded animals.;
申请公布号 US9357782(B2) 申请公布日期 2016.06.07
申请号 US201314418100 申请日期 2013.08.06
申请人 NOVARTIS TIERGESUNDHEIT AG 发明人 Gauvry Noelle;Pautrat Francois
分类号 C07D239/48;C07D401/14;C07D403/14;A01N43/54;A01N43/90;C07D403/12;C07D413/14;C07D213/74;C07D401/04;C07D401/12;C07D403/04;C07D239/47;C07D487/10;A01N43/60;A01N43/62;A01N43/84 主分类号 C07D239/48
代理机构 代理人 McGraw Elizabeth A.
主权项 1. The compound of formula Ia wherein one of R1 and R1′ is H and the other one is H, halogen, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-alkylthio, or amino, N-mono- or N,N-di-C1-C4-alkylamino; x and y are each independently of the other 1, 2 or 3; R2 and R3 are each independently of the other halogen, cyano, nitro, C1-C4-alkyl, C1-C2-haloalkyl, C1-C2-alkoxy, C1-C2-haloalkoxyl, C1-C2-alkylthio, C1-C2-haloalkylthio, C1-C2-alkylsulfonyl, halo-C1-C2-alkylsulfonyl, amino, N-mono- and N,N-di-C1-C4-alkylamino, aminosulfonyl and C1-C2-alkylaminosulfonyl; wherein, if x or y is 2 or 3, the two or three radicals R2 or R3 each may be same or different; L1 is a radical of formula wherein X1, X2 and X3 are each independently NH, N(C1-C2-alkyl) or O, Y is —CH2—, —NH—, —C(O)— or —S(O2)—, p″ is 0 or 1 r′ is 0, 1 or 2, r and s are each independently 1 or 2, s′ is an integer 0, 1 or 2; and A3 is C2-C4-alkylene or C3-C6-cycloalkylene; and L2 is a radical of formula wherein Y is —CH2—, —NH—, —C(O)— or —S(O)2—, t is 0 or 1, and X5 and X6 are each independently O or NH or N(CH3).
地址 Basel CH