发明名称 A PROCESS FOR PREPARING 7-[(3R)-3-AMINO-L-OXO-4-(2,4,5TRIFLUOROPHENYL)BUTYI]- 5,6,7,8-TETRAHYDRO-3-(TRIFLUOROMETHYL)-L,2,4-TRIAZOLO[4,3-A]PYRAZINE HYDROCHLORIDE MONOHYDRATE AND ITS CRYSTALLINE FORM
摘要 The present invention discloses industrially feasible process for preparation of 7-[(3R)-3- amino-l-oxo-4-(2,4,5trifluorophenyl)butyl]-5,6,7,8-tetrahydro-3-(trifluorornethyl)-l,2,4- triazolo[4,3-a]pyrazine Hydrochloride monohydrate.
申请公布号 WO2016162877(A1) 申请公布日期 2016.10.13
申请号 WO2015IN00328 申请日期 2015.08.24
申请人 HARMAN FINOCHEM LIMITED 发明人 HARMAN FINOCHEM LIMITED;KADAM, Vijay Trimbak;SARANAPU, Nareesh;SINGAMPALLLI, Sri Hari;MINHAS, Harpreet Singh;MINHAS, Gurpreet Singh
分类号 C07D487/04 主分类号 C07D487/04
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