发明名称 AZACARBAZOLE BTK INHIBITORS
摘要 The present invention provides Bruton's Tyrosine Kinase (Btk) inhibitor compounds according to Formula (I), or pharmaceutically acceptable salts thereof, wherein CH, R1, R1a, R1b, R2, R3, and the subscripts m1, m2, p, q, and t are as set forth herein. The present invention also provides pharmaceutical compositions comprising these compounds and their use in therapy. In particular, the present invention relates to the use of Btk inhibitor compounds of Formula (I) in the treatment of Btk mediated disorders.
申请公布号 WO2016164284(A1) 申请公布日期 2016.10.13
申请号 WO2016US25808 申请日期 2016.04.04
申请人 MERCK SHARP & DOHME CORP.;LIU, Jian;KOZLOWSKI, Joseph;KIM, Ronald;GAO, Xiaolei;BOGA, Sobhana Babu;YU, Younong;WU, Hao;LIU, Shilan;YANG, Chundao 发明人 LIU, Jian;KOZLOWSKI, Joseph;KIM, Ronald;GAO, Xiaolei;BOGA, Sobhana Babu;YU, Younong;WU, Hao;LIU, Shilan;YANG, Chundao
分类号 A61K31/5377;A61K31/541;A61K31/55;C07D487/04 主分类号 A61K31/5377
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