发明名称 CRYSTALLINE SOLVATES AND COMPLEXES OF (1S)-1,5-ANHYDRO-1-C-(3-((PHENYL)METHYL)PHENYL-D-GLUCITOL DERIVATIVES WITH AMINO ACIDS AS SGLT2 INHIBITORS FOR THE TREATMENT OF DIABETES
摘要 The present invention relates to physical crystal structures of a compound of the formula I: wherein R1, R2, R2a, R3 and R4 are as defined herein, especially pharmaceutical compositions containing structures of compound I or II, processes for preparing same, intermediates used in preparing same, and methods of treating diseases such as diabetes using such structures.
申请公布号 CA2653344(C) 申请公布日期 2016.06.07
申请号 CA20072653344 申请日期 2007.06.21
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 GOUGOUTAS, JACK Z.;LOBINGER, HILDEGARD;RAMAKRISHNAN, SRIVIDYA;DESHPANDE, PRASHANT P.;BIEN, JEFFREY T.;LAI, CHIAJEN;WANG, CHENCHI;RIEBEL, PETER;GROSSO, JOHN ANTHONY;NIRSCHL, ALEXANDRA A.;SINGH, JANAK;DIMARCO, JOHN D.
分类号 C07H7/04;A61K31/351;A61P3/06;A61P3/10;A61P5/50 主分类号 C07H7/04
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