发明名称 1-Aryl-5-alkyl pyrazole derivative compounds, processes of making and methods of using thereof
摘要 Provided are 1-aryl-5-alkyl pyrazole compounds, of formula (I): wherein: R<SUB>1 </SUB>is hydrogen, cyano, halogen, R<SUB>8</SUB>, formyl, -C(O)R<SUB>8</SUB>, -C(O)OR<SUB>8</SUB>, -C(O)NR<SUB>9</SUB>R<SUB>10</SUB>, or -C(S)NH<SUB>2</SUB>; R<SUB>2 </SUB>is R<SUB>2 </SUB>or -S(O)<SUB>m</SUB>R<SUB>11</SUB>; R<SUB>3 </SUB>is methyl, ethyl or C<SUB>1</SUB>-C<SUB>4 </SUB>haloalkyl; R<SUB>4</SUB>, R<SUB>5 </SUB>and R<SUB>7 </SUB>are independently hydrogen, halogen, alkyl, haloalkyl, cyano or nitro; R<SUB>6 </SUB>is halogen, alkyl, haloalkyl, alkoxy, haloalkyloxy, cyano, nitro, -C(O)R<SUB>12</SUB>, -S(O)<SUB>n</SUB>R<SUB>12 </SUB>or SF<SUB>5</SUB>; Z is a nitrogen atom or C-R<SUB>13</SUB>; R<SUB>8 </SUB>is alkyl, haloalkyl, cycloalkyl or halocycloalkyl; R<SUB>9 </SUB>is hydrogen, alkyl, haloalkyl or alkoxy; R<SUB>10 </SUB>is hydrogen, alkyl, haloalkyl or alkoxy; R<SUB>11 </SUB>is alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl or cycloalkyl; R<SUB>12 </SUB>is alkyl or haloalkyl; R<SUB>13 </SUB>is hydrogen, halogen, cyano, nitro, alkyl, haloalkyl, alkoxy or haloalkoxy; m is 0, 1 or 2; and n is 0, 1 or 2; or a salt thereof, the method of making compounds of formula (I) and the use of these compounds against ectoparasites, endoparasites and pests.
申请公布号 US2008031902(A1) 申请公布日期 2008.02.07
申请号 US20070825050 申请日期 2007.07.03
申请人 发明人 LEE HYOUNG I.;DE FALLOIS LOIC P.L.;TIMMONS PHILIP R.;CAWTHORNE WILLIAM G.JR.;DE LEON ADALBERTO P.
分类号 A01N25/00;A01N43/56;A01P15/00;C07D231/10;C07D231/16 主分类号 A01N25/00
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