发明名称 Benzimidazole-carboxamide compounds as 5-HT4 receptor agonists
摘要 The invention relates to benzimidazole-carboxamide 5-HT4 receptor agonist compounds of formula (I) wherein R1 and X are as defined in the specification, or a pharmaceutically acceptable salt or solvate or stereoisomer thereof. The invention also relates to pharmaceutical compositions comprising such compounds, methods of using such compounds to treat diseases associated with 5-HT4 receptor activity, and processes and intermediates useful for preparing such compounds. The invention further relates to crystalline forms of a compound of formula (I).
申请公布号 US8143279(B2) 申请公布日期 2012.03.27
申请号 US20060920817 申请日期 2006.05.24
申请人 MCKINNELL ROBERT MURRAY;LONG DANIEL D.;DALZIEL SEAN;PHIZACKERLEY KIRSTEN M.;THERAVANCE, INC. 发明人 MCKINNELL ROBERT MURRAY;LONG DANIEL D.;DALZIEL SEAN;PHIZACKERLEY KIRSTEN M.
分类号 A61K31/4545;C07D403/14 主分类号 A61K31/4545
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