发明名称 HETEROBICYCLES FKBP-LIGANDS
摘要 Diazabicyclo[3.3.1]nonane derivatives that inhibit the peptidyl-prolyl isomerase enzyme activity associated with FK-506 binding proteins (FKBP) are described for treating neurological disorders. Also described are compounds useful for preparing such inhibitors.
申请公布号 WO02089806(A1) 申请公布日期 2002.11.14
申请号 WO2002US14966 申请日期 2002.05.10
申请人 AGOURON PHARMACEUTICALS, INC.;GUO, CHUANGXING;AUGELLI-SZAFRAN, CORINNE, E.;BARTA, NANCY, SUE;BENDER, STEVEN, LEE;BIGGE, CHRISTOPHER, FRANKLIN;CAPRATHE, BRADLEY, WILLIAM;CHATTERJEE, ARINDAM;DEAL, JUDITH;DONG, LIMING;FAY, LORRAINE, KATHLEEN;HOU, XINJUN;HUDACK, RAYMOND, ANDREW, JR.;WARNER-LAMBERT COMPANY 发明人 GUO, CHUANGXING;AUGELLI-SZAFRAN, CORINNE, E.;BARTA, NANCY, SUE;BENDER, STEVEN, LEE;BIGGE, CHRISTOPHER, FRANKLIN;CAPRATHE, BRADLEY, WILLIAM;CHATTERJEE, ARINDAM;DEAL, JUDITH;DONG, LIMING;FAY, LORRAINE, KATHLEEN;HOU, XINJUN;HUDACK, RAYMOND, ANDREW, JR.;WARNER-LAMBERT COMPANY
分类号 C07D451/14;A61K31/439;A61K31/4995;A61K31/5365;A61K31/5377;A61P9/10;A61P17/14;A61P21/02;A61P25/00;A61P25/16;A61P25/28;A61P27/02;A61P27/16;A61P43/00;C07C57/58;C07C59/64;C07D471/08;C07D471/18;C07D498/18;C07D519/00;(IPC1-7):A61K31/499;A61K31/536;C07C59/68;C07C233/65;C07C235/46 主分类号 C07D451/14
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