发明名称 METHOD FOR PRODUCING 5-HYDROXYPIPERIDINE-2-CARBOXYLIC ACID
摘要 A method for producing (2 S ,5 S )/(2 R ,5 R )-5-hydroxypiperidine-2-carboxylic acid represented by the formula (10) below: , the method comprising the step of removing the protecting group from the hydroxyl group in a compound represented by the formula (7) below: (wherein P represents a protecting group, R 3 represents an alkyl group containing 1 to 4 carbon atoms, and A represents an alkyl group containing 1 to 10 carbon atoms, an aryl group containing 6 to 12 carbon atoms, an alkyloxy group containing 1 to 4 carbon atoms, or an aralkyloxy group containing 7 to 20 carbon atoms) to synthesize a compound represented by the formula (8) below: (wherein R 3 represents an alkyl group containing 1 to 4 carbon atoms, and A represents an alkyl group containing 1 to 10 carbon atoms, an aryl group containing 6 to 12 carbon atoms, an alkyloxy group containing 1 to 4 carbon atoms, or an aralkyloxy group containing 7 to 20 carbon atoms).
申请公布号 EP3091002(A1) 申请公布日期 2016.11.09
申请号 EP20140873766 申请日期 2014.12.26
申请人 API CORPORATION 发明人 TAKEHARA, JUN;MURAI, MASATO;OHTANI, TAKASHI;MAEDA, TOMOKO;HIDAKA, TSUGIHIKO
分类号 C07D211/60;C07B61/00;C07C233/47;C07C309/66;C07D498/08 主分类号 C07D211/60
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