发明名称 |
9-(ARYL OR HETEROARYL)-2-(PYRAZOLYL, PYRROLIDINYL OR CYCLOPENTYL)AMINOPURINE DERIVATIVES AS ANTICANCER AGENTS |
摘要 |
Compounds of the formula I in which X, R1 and R2 have the meanings indicated in Claim 1, are inhibitors of GCN2, and can be employed, inter alia, for the treatment of cancer. |
申请公布号 |
EP2964648(B1) |
申请公布日期 |
2016.11.16 |
申请号 |
EP20140705029 |
申请日期 |
2014.02.11 |
申请人 |
MERCK PATENT GMBH |
发明人 |
HOELZEMANN, GUENTER;DORSCH, DIETER;WEGENER, ANSGAR;POESCHKE, OLIVER;BUSCH, MICHAEL;SEENISAMY, JEYAPRAKASHNARAYANAN |
分类号 |
C07D473/32;A61K31/52;A61P35/00 |
主分类号 |
C07D473/32 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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