发明名称 |
3-ARYL-4-AMIDO-BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS |
摘要 |
The present disclosure relates to inhibitors of zinc-dependent histone deacetylases (HDACs) useful in the treatment of diseases or disorders associated with an HDAC, e.g., HDAC6, having a Formula I:(Formula I should be inserted here) where R, L, X1, X2, X3, X4, Y1, Y2, Y3, and Y4 are described herein. |
申请公布号 |
WO2016126724(A1) |
申请公布日期 |
2016.08.11 |
申请号 |
WO2016US16200 |
申请日期 |
2016.02.02 |
申请人 |
FORMA THERAPEUTICS, INC. |
发明人 |
ZHENG, XIAOZHANG;NG, PUI YEE;HAN, BINGSONG;THOMASON, JENNIFER R.;ZABLOCKI, MARY-MARGARET;LIU, CUIXIAN;DAVIS, HEATHER;RUDNITSKAYA, ALEKSANDRA;LANCIA JR., DAVID;MILLAN, DAVID S.;MARTIN, MATTHEW W. |
分类号 |
C07D403/06;A61K31/551;A61K31/553;A61P35/00;C07D243/14;C07D267/12;C07D413/06 |
主分类号 |
C07D403/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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