发明名称 3-ARYL-4-AMIDO-BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
摘要 The present disclosure relates to inhibitors of zinc-dependent histone deacetylases (HDACs) useful in the treatment of diseases or disorders associated with an HDAC, e.g., HDAC6, having a Formula I:(Formula I should be inserted here) where R, L, X1, X2, X3, X4, Y1, Y2, Y3, and Y4 are described herein.
申请公布号 WO2016126724(A1) 申请公布日期 2016.08.11
申请号 WO2016US16200 申请日期 2016.02.02
申请人 FORMA THERAPEUTICS, INC. 发明人 ZHENG, XIAOZHANG;NG, PUI YEE;HAN, BINGSONG;THOMASON, JENNIFER R.;ZABLOCKI, MARY-MARGARET;LIU, CUIXIAN;DAVIS, HEATHER;RUDNITSKAYA, ALEKSANDRA;LANCIA JR., DAVID;MILLAN, DAVID S.;MARTIN, MATTHEW W.
分类号 C07D403/06;A61K31/551;A61K31/553;A61P35/00;C07D243/14;C07D267/12;C07D413/06 主分类号 C07D403/06
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