发明名称 |
LOWCOST, HIGH YIELD SYNTHESIS OF NEVIRAPINE |
摘要 |
Improved methods of producing the HIV drug substance, nevirapine are provided. The methods employ a cost effective and high yield synthetic methods for preparing the nevirapine building block 2-chloro-3-amino-4-picoline (CAPIC) and 2-cyclopropyl amino nicotinate (Me-CAN), and improvements in other steps of nevirapine synthesis. |
申请公布号 |
WO2016118586(A1) |
申请公布日期 |
2016.07.28 |
申请号 |
WO2016US14066 |
申请日期 |
2016.01.20 |
申请人 |
VIRGINIA COMMONWEALTH UNIVERSITY |
发明人 |
AHMAD, SAEED;GUPTON, FRANK;VERGHESES, JENSON;MCQUADE, TYLER |
分类号 |
C07D213/73 |
主分类号 |
C07D213/73 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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