发明名称 MACROCYCLIC DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES
摘要 Compound of formula (I), which substitute A is selected from C6-C12 aryl and 5-6 member heteroaryl, and values of R2, R3, R4, X, Y, Z and n, m, p substitudes are provided in the claims or their pharmaceutically acceptable salt, and composition on basis thereof; application of said compound or salt therefor cancer treating medicine preparation. Tables: 1
申请公布号 GEP201606560(B) 申请公布日期 2016.10.25
申请号 GE2013AP13564 申请日期 2013.02.20
申请人 PFIZER INC 发明人 BAILEY, SIMON;BURKE, BENJAMIN, JOSEPH;COLLINS, MICHAEL, RAYMOND;CUI, JINGRONG, JEAN;DEAL, JUDITH, GAIL;HOFFMAN, ROBERT, LOUIS;HUANG, QINHUA;JOHNSON, TED, WILLIAM;KANIA, ROBERT, STEVEN;KATH, JOHN, CHARLES;LE, PHUONG, THI, QUY;MCTIGUE, MICHELE, ANN;PALMER, CYNTHIA, LOUISE;RICHARDSON, PAUL, FRANCIS;SACH, NEAL, WILLIAM
分类号 C07D491/08;A61K31/4353;C07D491/18;C07D498/08;C07D498/18;C07D498/22;C07D513/18 主分类号 C07D491/08
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