发明名称 PHARMACEUTICAL COMPOSITIONS CONTAINING SULPHONIC ACID DERIVATIVES
摘要 A naphthalenesulfonic acid or quinolinesulfonic acid of formula (I), wherein A is N or a CR8 formula group, where R8 is H, OH, NR10OR11, independently from one another, where R10 and R11 represent H or C1-C6 alkyl or a group of formula NH-CO-R12, where R12 is C1-C6 alkyl or C6-C10 aryl; R1 and R2 represent H or SO3R9, independently from one another, where R9 is H, ammonium or a cation of an alkali or alkaline-earth metal; R3 is H or OH; and R4, R5, R6 and R7 represent H, an NR10R11 or NH-CO-R12 group, independently from one another; on the condition that (i) at least one of R1 or R2 is SO3R9, and (ii) at least one of R4, R5, R6 or R7 is an NR10R11 or NH-CO-R12 group, or their pharmaceutically acceptable salts; and a pharmaceutically acceptable excipient.
申请公布号 US2009076140(A1) 申请公布日期 2009.03.19
申请号 US20080264000 申请日期 2008.11.03
申请人 ITALFARMACO, S. A.;CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS;INSTITUTO MADRILENO DE LA SALUD 发明人 BANFI TOSI BEATRIZ MARIA;GIMENEZ GALLEGO GUILLERMO;VALVERDE LOPEZ SERAFIN;LOZANO PUERTO ROSA MARIA;SANCHEZ CUEVAS PEDRO
分类号 A61K31/255;A61K31/185;A61K31/47;A61P3/04;A61P9/10;A61P17/06;A61P19/02 主分类号 A61K31/255
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