发明名称 |
PHARMACEUTICAL FORMULATIONS COMPRISING A PYRIDYLAMINOACETIC ACID COMPOUND |
摘要 |
Provided is a pharmaceutical preparation for treatment or prevention of glaucoma or ocular hypertension, comprising 0.0003 to 0.01% (w/v) of isopropyl (6-{[4-(pyrazol-1-yl)benzyl] (pyridin-3-ylsulfonyl)aminomethyl}pyridin-2-ylamino) acetate, or a salt thereof. The pharmaceutical preparation has an excellent intraocular pressure lowering effect and may be used as a therapeutic or preventive agent for glaucoma or ocular hypertension or an intraocular pressure lowering agent. |
申请公布号 |
US2016324838(A1) |
申请公布日期 |
2016.11.10 |
申请号 |
US201615212592 |
申请日期 |
2016.07.18 |
申请人 |
SANTEN PHARMACEUTICAL CO., LTD. |
发明人 |
SHAMS Naveed;KROON Henk-Andre;KAWATA Hisashi;KAWABATA Noriko |
分类号 |
A61K31/444;A61K9/00 |
主分类号 |
A61K31/444 |
代理机构 |
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代理人 |
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主权项 |
1. A pharmaceutical preparation for treatment or prevention of glaucoma or ocular hypertension, comprising 0.001 to 0.01% (w/v) of isopropyl (6-{[4-(pyrazol-1-yl)benzyl] (pyridin-3-ylsulfonyl) aminomethyl}pyridin-2-ylamino) acetate, or a salt thereof. |
地址 |
Osaka JP |