发明名称 |
PROCESS FOR PREPARATION OF 2-ALKOXY-5-(PYRIDIN-2-YL)PYRIDINE AS INTERMEDIATE OF PERAMPANEL |
摘要 |
<P>PROBLEM TO BE SOLVED: To provide an alternative process for preparation of 2-alkoxy-5-(pyridin-2-yl)pyridine or a salt thereof, making it possible to overcome at least partially the drawbacks of the conventional technology. <P>SOLUTION: There is provided a process for synthesis of 2-alkoxy-5-(pyridin-2-yl)pyridine which is an intermediate for the synthesis of the active substance perampanel. <P>COPYRIGHT: (C)2013,JPO&INPIT |
申请公布号 |
JP2013095752(A) |
申请公布日期 |
2013.05.20 |
申请号 |
JP20120230411 |
申请日期 |
2012.10.18 |
申请人 |
FIS FABBRICA ITALIANA SINTETICI SPA |
发明人 |
FONTANA FRANCESCO;STABILE PAOLO |
分类号 |
C07D213/64;A61K31/444;A61P25/00;A61P25/08;A61P25/16;C07B61/00;C07F3/02 |
主分类号 |
C07D213/64 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|