发明名称 PROCESS FOR PREPARATION OF 2-ALKOXY-5-(PYRIDIN-2-YL)PYRIDINE AS INTERMEDIATE OF PERAMPANEL
摘要 <P>PROBLEM TO BE SOLVED: To provide an alternative process for preparation of 2-alkoxy-5-(pyridin-2-yl)pyridine or a salt thereof, making it possible to overcome at least partially the drawbacks of the conventional technology. <P>SOLUTION: There is provided a process for synthesis of 2-alkoxy-5-(pyridin-2-yl)pyridine which is an intermediate for the synthesis of the active substance perampanel. <P>COPYRIGHT: (C)2013,JPO&INPIT
申请公布号 JP2013095752(A) 申请公布日期 2013.05.20
申请号 JP20120230411 申请日期 2012.10.18
申请人 FIS FABBRICA ITALIANA SINTETICI SPA 发明人 FONTANA FRANCESCO;STABILE PAOLO
分类号 C07D213/64;A61K31/444;A61P25/00;A61P25/08;A61P25/16;C07B61/00;C07F3/02 主分类号 C07D213/64
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