发明名称 |
BICYCLIC NITROGENOUS FUSED-RING COMPOUND |
摘要 |
A novel compound having an excellent antagonistic effect on a corticotropin-releasing-factor receptor. It is a compound represented by the following formula or a salt thereof. (I) In the formula, R<1> represents hydrogen, C1-6 alkyl, C1-6 alkoxy, etc.; R<2> represents halogeno, cyano, nitro, C1-10 alkyl, C2-10 alkenyl, C2-10 alkynyl, etc.; R<3> represents an optionally substituted C6-14 aromatic hydrocarbon group or an optionally substituted, 5- to 14-membered aromatic heterocyclic group; and X, Y, and Z each independently represents nitrogen or CR<4> (wherein R<4> represents hydrogen, halogeno, cyano, nitro, optionally halogenated C1-6 alkyl, etc.), provided that at least two of X, Y, and Z represent CR<4>.
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申请公布号 |
WO02062800(A1) |
申请公布日期 |
2002.08.15 |
申请号 |
WO2002JP01098 |
申请日期 |
2002.02.08 |
申请人 |
EISAI CO., LTD.;HIBI, SHIGEKI;TAKAHASHI, YOSHINORI;HOSHINO, YORIHISA;KIKUCHI, KOICHI;SOEJIMA, MOTOHIRO;YOSHIUCHI, TATSUYA;SHIN, KOGYOKU;ONO, MUTSUKO;SHIBATA, HISASHI;INO, MITSUHIRO;HIRAKAWA, TETSUYA |
发明人 |
HIBI, SHIGEKI;TAKAHASHI, YOSHINORI;HOSHINO, YORIHISA;KIKUCHI, KOICHI;SOEJIMA, MOTOHIRO;YOSHIUCHI, TATSUYA;SHIN, KOGYOKU;ONO, MUTSUKO;SHIBATA, HISASHI;INO, MITSUHIRO;HIRAKAWA, TETSUYA |
分类号 |
A61P1/14;A61P3/04;A61P3/10;A61P9/00;A61P9/02;A61P9/06;A61P9/10;A61P9/12;A61P11/00;A61P11/06;A61P13/00;A61P15/08;A61P15/10;A61P15/12;A61P17/14;A61P19/10;A61P21/00;A61P21/02;A61P25/00;A61P25/02;A61P25/04;A61P25/06;A61P25/08;A61P25/20;A61P25/28;A61P25/30;A61P25/32;A61P27/00;A61P27/06;A61P29/00;A61P31/18;A61P35/00;A61P37/04;A61P37/08;A61P43/00;C07D471/04;C07D487/04;(IPC1-7):C07D487/04;A61K31/498;A61K31/502;A61K31/537;A61K31/437;A61K31/519 |
主分类号 |
A61P1/14 |
代理机构 |
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代理人 |
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地址 |
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