发明名称 BENZOIMIDAZOL-2-YL PYRIMIDINE MODULATORS OF THE HISTAMINE H4 RECEPTOR
摘要 Benzoimidazol-2-yl pyrimidines, purification methods for the same, and pharmaceutical compositions and methods for the treatment of disease states, disorders, and conditions mediated by H4 receptor activity, including allergy, asthma, autoimmune diseases, and pruritus.
申请公布号 US2016159775(A1) 申请公布日期 2016.06.09
申请号 US201615047359 申请日期 2016.02.18
申请人 Janssen Pharmaceutica NV 发明人 Conza Matteo;Hickey Magali B.;Horns Stefan;Lochner Susanne
分类号 C07D401/14;C30B7/08;C30B29/54;C07C51/43 主分类号 C07D401/14
代理机构 代理人
主权项 1. A hemitartrate tetrahydrate of [5-(4,6-Dimethyl-1H-benzoimidazol-2-yl)-4-methyl-pyrimidin-2-yl]-[3-(1-methyl-piperidin-4-yl)-propyl]-amine of formula:
地址 Beerse BE
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