发明名称 |
PHOSPHONOOXY QUINAZOLINE DERIVATIVE AND ITS PHARMACEUTICAL USE |
摘要 |
<p><P>PROBLEM TO BE SOLVED: To provide a new antitumor agent. <P>SOLUTION: The antitumor agent is 2-[[3-(ä4-[(5-ä2-[(3-fluorophenyl)amino]-2-oxoethyl}-1H-pyrazol-3-yl)amino]-quinazolin-7-yl}oxy)propyl](ethyl)amino]ethyl dihydrogenphosphate or a pharmaceutically acceptable salt thereof. A pharmaceutical composition containing the same and its therapeutic use are also provided. <P>COPYRIGHT: (C)2009,JPO&INPIT</p> |
申请公布号 |
JP2009046514(A) |
申请公布日期 |
2009.03.05 |
申请号 |
JP20080265949 |
申请日期 |
2008.10.15 |
申请人 |
ASTRAZENECA AB |
发明人 |
HERON NICOLA MURDOCH;JUNG FREDERIC HENRI;PASQUET GEORGES RENE;MORTLOCK ANDREW AUSTEN |
分类号 |
C07F9/6512;A61K31/661;A61K31/675;A61P35/00;A61P35/02;A61P43/00;C07D401/14;C07D403/12;C07D403/14;C07F9/6558 |
主分类号 |
C07F9/6512 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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