发明名称 PROCESS AND INTERMEDIATES FOR THE PREPARATION OF THE THIENOPYRROLE DERIVATIVES
摘要 <p>A process for preparing a compound of formula (I) where R4 and R5are as defined in the specification; and R6 is hydrogen or a protecting group, which process comprises cyclisation of a compound of formula (II) where R 4, R5and R6 are as defined in relation to formula (I) and R7is a nitrogen-protecting group, and removing protecting group R7-, and thereafter if desired or necessary, removing any protecting group R6 to obtain the corresponding carboxylic acid. Novel intermediates and the use of the products in the preparation of pharmaceutical compounds is also described and claimed.</p>
申请公布号 KR20050061503(A) 申请公布日期 2005.06.22
申请号 KR20057005618 申请日期 2005.03.31
申请人 ASTRAZENECA AB 发明人 PARKER JEREMY STEPHEN;SCHOFIELD PAUL;STOCKER ANDREW;MURRAY PAUL MICHAEL
分类号 C07D333/36;C07D495/04;(IPC1-7):C07D495/04 主分类号 C07D333/36
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