发明名称 |
Melanocortin receptor ligands |
摘要 |
The present invention relates to compounds which comprise a 4-substituted piperidine ring linked to a substituted or unsubstituted hydrocarbyl ring. The compounds, including all enatiomeric and diasteriomeric forms and pharmaceutically acceptable salts thereof, have the formula: wherein preferably R is substituted aryl, W is a pendant unit having the formula: <?in-line-formulae description="In-line Formulae" end="lead"?>-L-Q <?in-line-formulae description="In-line Formulae" end="tail"?> L is a linking unit, Q is preferably a cyclic hydrocarbyl unit; W<SUP>1 </SUP>is preferably a carbocyclic unit and W<SUP>2 </SUP>is a heteroatom comprising unit.
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申请公布号 |
US2005171158(A1) |
申请公布日期 |
2005.08.04 |
申请号 |
US20050092100 |
申请日期 |
2005.03.29 |
申请人 |
EBETINO FRANK H.;LIU XUEWEI;SOLINSKY MARK G.;WOS JOHN A. |
发明人 |
EBETINO FRANK H.;LIU XUEWEI;SOLINSKY MARK G.;WOS JOHN A. |
分类号 |
C07D211/16;A61K31/445;A61K31/454;A61K31/4545;A61P1/14;A61P1/16;A61P3/04;A61P3/06;A61P3/08;A61P3/10;A61P5/24;A61P7/00;A61P7/02;A61P9/10;A61P9/12;A61P11/00;A61P15/00;A61P15/10;A61P19/02;A61P19/06;A61P21/02;A61P25/00;A61P29/00;A61P31/10;A61P35/00;C07D211/26;C07D211/58;C07D401/06;C07D401/14;(IPC1-7):A61K31/445;C07D211/06;C07D41/02 |
主分类号 |
C07D211/16 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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