发明名称 NOVEL CRYSTALLINE FORM B OF CARVEDILOL DIHYDROGEN PHOSPHATE
摘要 <p>A novel crystalline form B of carvedilol dihydrogen phosphate having X-ray diffraction pattern as shown in figure 1. A process for the preparation of crystalline form B of carvedilol dihydrogen phosphate according to claim 1 that comprises dissolving carvedilol base in aprotic polar solvent, addition of phosphoric acid, heating the solution, adding water to hot solution, cooling, and isolation of solid.</p>
申请公布号 WO2009008009(A4) 申请公布日期 2009.03.05
申请号 WO2008IN00441 申请日期 2008.07.09
申请人 LUPIN LIMITED;THAPER, RAJESH, KUMAR;PRABHAVAT, MANOJ, DEVILALJI;MOUNISHWARACHAR, A., V.;PAWAR, YOGESH, DADAJI;UPADHAY, PRITESH, R. 发明人 THAPER, RAJESH, KUMAR;PRABHAVAT, MANOJ, DEVILALJI;MOUNISHWARACHAR, A., V.;PAWAR, YOGESH, DADAJI;UPADHAY, PRITESH, R.
分类号 C07D209/88;A61K31/403;A61P9/12 主分类号 C07D209/88
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