发明名称 SERINE/THREONINE KINASE INHIBITORS.
摘要 Compounds having the formula I wherein R1, X1, X2, X3 and X4 as defined herein are inhibitors of ERK kinase. Also disclosed are compositions and methods for treating hyperproliferative disorders.
申请公布号 MX2016007352(A) 申请公布日期 2016.09.08
申请号 MX20160007352 申请日期 2014.12.03
申请人 GENENTECH, INC. 发明人 DO, Steven;KOLESNIKOV, Aleksandr
分类号 C07D498/16;A61K31/4353;C07D471/16 主分类号 C07D498/16
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