发明名称 PYRROLO[2,3-D]PYRIMIDINYL, PYRROLO[2,3-B]PYRAZINYL AND PYRROLO[2,3-D]PYRIDINYL ACRYLAMIDES.
摘要 The present invention provides pharmaceutically active pyrrolo[2,3- d]pyrimidinyl and pyrrolo[2,3-d]pyridinyl acrylamides and analogues thereof. Such compounds are useful for inhibiting Janus Kinase (JAK). This invention also is directed to compositions comprising methods for making such compounds, and methods for treating and preventing conditions mediated by JAK.
申请公布号 MX2016007156(A) 申请公布日期 2016.07.21
申请号 MX20160007156 申请日期 2014.11.20
申请人 PFIZER INC. 发明人 MATTHEW MERRILL HAYWARD;ATLI THORARENSEN;MATTHEW FRANK BROWN;AGUSTIN CASIMIRO-GARCIA;YE CHE;JOTHAM WADSWORTH COE;MARK EDWARD FLANAGAN;ADAM MATTHEW GILBERT;JONATHAN DAVID LANGILLE;JUSTIN IAN MONTGOMERY;JEAN- BAPTISTE TELLIEZ;RAYOMAND JAL UNWALLA;JOHN I. TRUJILLO
分类号 C07D471/04;A61K31/4375;A61P35/00;C07D487/04 主分类号 C07D471/04
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