发明名称 Substituted benzoxazoles and analogues as estrogenic agents
摘要 This invention provides estrogen receptor modulators of formula I, having the structure wherein R 1 , R 2 , R 2a , R 3 , R 3a , and R 4 , and X as defined in the specification, or a pharmaceutically acceptable salt thereof for the treatment of inflammatory bowel diseases.
申请公布号 ZA200405249(B) 申请公布日期 2007.01.31
申请号 ZA20040005249 申请日期 2004.07.01
申请人 WYETH 发明人 MALAMAS, MICHAEL SOTIRIOS;GUNAWAN, IWAN;COLLINI, MICHAEL DAVID;KEITH, JR., JAMES CARL;LYTTLE, CECIL RICHARD;MCDEVITT, ROBERT EMMETT;MANAS, ERIC STEVEN;HARRIS, HEATHER ANNE;ALBERT, LEO MASSILLAMONEY
分类号 C07D263/56;A61K;A61K31/423;A61K31/427;A61P;A61P1/04;A61P3/06;A61P3/10;A61P5/30;A61P5/32;A61P7/00;A61P9/00;A61P9/10;A61P9/12;A61P11/06;A61P13/00;A61P13/02;A61P13/08;A61P15/00;A61P17/02;A61P19/02;A61P25/00;A61P25/22;A61P25/28;A61P29/00;A61P35/00;C07D;C07D235/18;C07D263/57;C07D277/66;C07D413/04;C07D417/04 主分类号 C07D263/56
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