发明名称 CRYSTALLINE FORMS OF ANTIVIRAL SOFOSBUVIR ANALOGUES
摘要 Crystalline solid forms of the anti-HCV compound (S)-isopropyl 2-((S)-(((2R,3R,4R,5R)-5-(2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-4-fluoro-3-hydroxy-4-methyltetrahydrofuran-2- yl)methoxy)(phenoxy)phosphorylamino)propanoate (Compound I) are described Also provided are processes of making and methods of using the crystalline forms.
申请公布号 EP3086795(A1) 申请公布日期 2016.11.02
申请号 EP20140819226 申请日期 2014.12.08
申请人 GILEAD PHARMASSET LLC 发明人 CASTEEL, MELISSA, JEAN;DASHNER, KATHLEEN;JUNG, HYUK-JUN;SEO, MUN, SIK;SHI, BING;WANG, FANG;ZIA, VAHID
分类号 A61K31/7072;A61P31/18;C07F9/6558;C07H19/10 主分类号 A61K31/7072
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