METHYL- AND TRIFLUOROMETHYL-SUBSTITUTED PYRROLOPYRIDINE INHIBITORS OF RORC2 AND METHODS OF USE THEREOF
摘要
The present invention provides methyl- and trifluoromethyl-substituted pyrrolopyridines, pharmaceutical compositions thereof, and uses thereof as RORC2 inhibitors.
申请公布号
CA2905407(A1)
申请公布日期
2016.03.26
申请号
CA20152905407
申请日期
2015.09.23
申请人
PFIZER INC.
发明人
FLICK, ANDREW CHRISTOPHER;JONES, PETER;KAILA, NEELU;MENTE, SCOT RICHARD;SCHNUTE, MARK EDWARD;TRZUPEK, JOHN DAVID;VAZQUEZ, MICHAEL L.;XING, LI;ZHANG, LIYING;WENNERSTAL, GORAN MATTIAS;ZAMARATSKI, EDOUARD