发明名称 AN IMPROVED PROCESS FOR THE PREPARATION OF SUBSTANTIALLY PURE AZILSARTAN
摘要 The present invention relates to an improved process for the preparation of substantially pure compound of 2-Ethoxy-1-[[2'-(2,5-dihydro-5-oxo-1,2,4-oxadiazol- 3-yl)biphenyl-4-yl]methyl]benzimidazole-7-carboxylic acid (Azilsartan) of Formula I, with a reduced content of desethyl impurity less than 0.1% and an efficient, commercially viable process for the preparation of pure intermediates of Azilsartan.
申请公布号 WO2016147120(A1) 申请公布日期 2016.09.22
申请号 WO2016IB51470 申请日期 2016.03.16
申请人 SMILAX LABORATORIES LIMITED;KOTAGIRI, Vijaya Kumar;YENUMULA, Raghavendra Rao;BANDARI, Mohan;SURYADEVARA, Murali Krishna 发明人 KOTAGIRI, Vijaya Kumar;YENUMULA, Raghavendra Rao;BANDARI, Mohan;SURYADEVARA, Murali Krishna
分类号 C07D235/26;C07D413/10 主分类号 C07D235/26
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