发明名称 |
COMPOUNDS FOR PREPARING IMMUNOLOGICAL ADJUVANT |
摘要 |
The present invention provides methods for preparing TLR-4 receptor agonist E6020:
and stereoisomers thereof, which compounds are useful as an immunological adjuvants when co-administered with antigens such as vaccines for bacterial and viral diseases. Also provided are synthetic intermediates. |
申请公布号 |
EP1910387(A1) |
申请公布日期 |
2008.04.16 |
申请号 |
EP20060785934 |
申请日期 |
2006.06.30 |
申请人 |
EISAI CO., LTD |
发明人 |
FANG, FRANCIS G.;FOY, JAMES E.;HAWKINS, LYNN;LEMELIN, CHARLES;LESCARBEAU, ANDRE;NIU, XIANG;WU, KUO-MING |
分类号 |
C07F9/09;C07C217/28;C07C271/16;C07D263/14;C07F9/141;C07F9/24 |
主分类号 |
C07F9/09 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|