发明名称 ERK INHIBITORS
摘要 The present invention provides a compound of Formula (I) or the pharmaceutically acceptable salts, esters, and prodrugs thereof, which are ERK2 inhibitors. The invention also provides a pharmaceutical composition comprising an effective amount of at least one compound of Formula (I) and a pharmaceutically acceptable carrier. The invention also provides a pharmaceutical composition comprising an effective amount of at least one compound of Formula (I) and an effective amount of at least one other pharmaceutically active ingredient (such as, for example, a chemotherapeutic agent), and a pharmaceutically acceptable carrier.
申请公布号 WO2016100050(A1) 申请公布日期 2016.06.23
申请号 WO2015US64860 申请日期 2015.12.10
申请人 MERCK SHARP & DOHME CORP.;SILIPHAIVANH, PHIENG;METHOT, JOEY;LIPFORD, KATHRYN ANN;MOLINARI, DANIELLE;SLOMAN, DAVID, L.;WITTER, DAVID;ZHOU, HUA;BOYCE, CHRISTOPHER;HUANG, XIANHAI;LIM, JONGWON;GUERIN, DAVID;KARUNAKARAN, GANESH BABU;BAKSHI, RAMAN KUMAR;LIU, ZIPING;FU, JIANMIN;WAN, ZHILONG;LIU, WEI 发明人 SILIPHAIVANH, PHIENG;METHOT, JOEY;LIPFORD, KATHRYN ANN;MOLINARI, DANIELLE;SLOMAN, DAVID, L.;WITTER, DAVID;ZHOU, HUA;BOYCE, CHRISTOPHER;HUANG, XIANHAI;LIM, JONGWON;GUERIN, DAVID;KARUNAKARAN, GANESH BABU;BAKSHI, RAMAN KUMAR;LIU, ZIPING;FU, JIANMIN;WAN, ZHILONG;LIU, WEI
分类号 C07D471/04 主分类号 C07D471/04
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