发明名称 A NEW PRODUCTION METHOD AND NEW INTERMEDIATES OF SYNTHESIS OF ELVITEGRAVIR
摘要 The present solution relates to an improved production method of elvitegravir of formula I, which is being clinically evaluated for treatment of HIV infection. Elvitegravir of formula I is produced via the intermediate of formula II, the preparation of which is also an object of the present solution.
申请公布号 EP2906529(B1) 申请公布日期 2016.11.23
申请号 EP20130782934 申请日期 2013.10.14
申请人 ZENTIVA, K.S. 发明人 RADL, STANISLAV
分类号 C07C227/10;C07C227/16;C07C229/34;C07D215/56 主分类号 C07C227/10
代理机构 代理人
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