| 发明名称 |
PYRAZOLE COMPOUNDS AS BTK INHIBITORS |
| 摘要 |
The present invention encompasses compounds of the formula (I) wherein the groups R1, Cy, and Y are defined herein, which are suitable for the treatment of diseases related to BTK, process of making, pharmaceutical preparations which contain compounds and their methods of use.; |
| 申请公布号 |
US2016340339(A1) |
申请公布日期 |
2016.11.24 |
| 申请号 |
US201515114923 |
申请日期 |
2015.01.23 |
| 申请人 |
Boehringer Ingelheim International GmbH |
发明人 |
BENTZIEN Joerg;BERRY Angela Kay;BOSANAC Todd;BURKE Michael Jason;DISALVO Darren Todd;MAO Can;MAO Wang;SHEN Yue |
| 分类号 |
C07D403/04;C07D401/04 |
主分类号 |
C07D403/04 |
| 代理机构 |
|
代理人 |
|
| 主权项 |
1. A compound of the formula (I) wherein R1 is H, C1-4 alkyl; Cy is chosen from wherein each phenyl or attached substituent thereof can be optionally substituted by halogen, —CN, haloalkyl, methyl, methoxy, hydroxyl; Y is a linker chosen from; R2 is chosen from or a pharmaceutically acceptable salt thereof. |
| 地址 |
Ingelheim am Rhein DE |
