发明名称 |
Alfa-form crystal of an acetanilide derivative |
摘要 |
To provide novel crystals useful as an ingredient for the production of a diabetes remedy. The invention is concerned with alpha -form crystal and beta -form crystal of (R)-2-(2-aminothiazol-4-yl)-4'-Ä2-Ä(2-hydroxy-2-phenylethyl)aminoÜethylÜacetanilide. The alpha -form crystal does not exhibit hygroscopicity and has stability such that it can be used as a medicine, and is useful for mass synthesis in the industrial production. The beta -form crystal does not relatively exhibit hygroscopicity and is also useful as a production intermediate of the alpha -form crystal. |
申请公布号 |
HU230481(B1) |
申请公布日期 |
2016.07.28 |
申请号 |
HU20040001665 |
申请日期 |
2002.10.29 |
申请人 |
ASTELLAS PHARMA INC. |
发明人 |
KAWAZOE SOUICHIROU;SAKAMOTO KENICHIROU;AWAMURA YUJI;MARUYAMA TATSUYA;SUZUKI TAKAYUKI;ONDA KENICHI;TAKASU TOSHIYUKI |
分类号 |
C07D277/40;A61K31/426;A61P3/10;C07D277/44 |
主分类号 |
C07D277/40 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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