发明名称 OXAZETIDINE DERIVATIVES, PROCESS FOR PREPARING THEM AND USE IN HUMAN MEDICINE AND IN COSMETICS
摘要 Compounds that are agonists of the MCIR receptor and that exhibit reduced toxicity relative to other compounds of the same class are described. These compounds can have the general formula (I) wherein: R1 represents a cyclopropylmethyl or a 4-hydroxybutyl group; R2 represents a hydrogen atom or a methyl group; and also the salts and enantiomers of the corresponding compounds of general formula (I). Also described, are methods for treating hypopigmentary pathologies and photosensitive dermatoses.
申请公布号 US2016237065(A1) 申请公布日期 2016.08.18
申请号 US201615139018 申请日期 2016.04.26
申请人 Galderma Research & Development 发明人 BOUIX-PETER Claire
分类号 C07D403/12;A61K8/49;A61Q5/00;A61K31/4178;A61Q19/08;A61Q19/00 主分类号 C07D403/12
代理机构 代理人
主权项 1. A compound of general formula (I) below: in which: R1 represents a cyclopropylmethyl or a 4-hydroxybutyl group; R2 represents a hydrogen atom or a methyl group; and also salts and enantiomers of the corresponding compounds of general formula (I).
地址 Biot FR