ANDROGEN RECEPTOR MODULATORS AND USES THEREOF

摘要

PROBLEM TO BE SOLVED: To provide novel androgen receptor modulators useful in treatment of cancer such as prostate cancer and a hormone dependent cancer.SOLUTION: The invention provides imidazolinone based compounds represented by formula (Ia) in the figure. [A is a pyridine ring; B is a benzene ring; X is O or S; two Rtogether form 1,3-propanediyl or the like; Rare independently -CH, -CF, OCHor the like; Rare independently H, halogen or the like; Ris -OCFor the like; m is 1, 2, 3 or 4; and n is 0, 1 or 2.]SELECTED DRAWING: None