发明名称 BENZOXABOROLE DERIVATIVES FOR TREATING BACTERIAL INFECTIONS
摘要 PROBLEM TO BE SOLVED: To provide a new broad spectrum of antimicrobials useful in combating microorganisms, especially those with multidrug resistance.SOLUTION: The present invention provides benzoxaborole compounds having structures represented by formula (I)-formula (III), or salts, hydrates or solvates thereof, particularly, the compounds preferably having (S) configuration in a configuration (Ris substituted/unsubstituted nitroalkyl or substituted/unsubstituted aminoalkyl; Ris halogen, unsubstituted alkyl, unsubstituted alkoxy or unsubstituted phenyl; Y is O or S; Ris substituted/unsubstituted alkyl or substituted/unsubstituted heteroalkyl).SELECTED DRAWING: None
申请公布号 JP2016199558(A) 申请公布日期 2016.12.01
申请号 JP20160114971 申请日期 2016.06.09
申请人 ANACOR PHARMACEUTICALS INC 发明人 HERNANDEZ VINCENT S;CHARLES DING;PLATTNER JACOB J;MICHAEL KEVIN RICHARD ALLEY;FERNANDO ROCK;ZHANG SUOMING;ERIC EASOM;LI XIANFENG;ZHOU DING
分类号 C07F5/04;A61K31/69;A61P31/04;A61P31/06;A61P43/00;C12Q1/04;C12Q1/48 主分类号 C07F5/04
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