发明名称 6-{8 {8 {8 (2-Cyanomethyl)amino{9 -1,2-dioxoethyl{9 -amino{9 acyl penicillins
摘要 6-[[[(2-Cyanomethyl)amino]-1,2-dioxoethyl]amino]acyl pencillins which have the formula <IMAGE> wherein R is hydrogen, lower alkyl, tri(lower alkyl)silyl, tri(lower alkyl)stannyl, trihaloethyl or a salt forming ion; R1 is hydrogen, lower alkyl, saturated or unsaturated cycloalkyl, phenyl, phenyl-lower alkyl, substituted phenyl or certain heterocyclic groups; R2 is hydrogen or methoxy; R3 is hydrogen, lower alkyl, phenyl-lower alkyl or cycloalkyl; and R4 and R5 each is hydrogen or lower alkyl, are useful as antibacterial agents.
申请公布号 US4168266(A) 申请公布日期 1979.09.18
申请号 US19780910546 申请日期 1978.05.30
申请人 E. R. SQUIBB & SONS, INC. 发明人 TREUNER, UWE D.;BREUER, HERMANN
分类号 C07D333/24;C07D499/00;C07D499/64;(IPC1-7):C07D499/64;C07D499/66;C07D499/68;C07D499/70 主分类号 C07D333/24
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