摘要 |
NEW MATERIAL:A pyridylalkyl N-(2,3-xylyl)anthranilate derivative expressed by the formula (R is 1-3C alkyl substituted by pyridyl group). EXAMPLE:2-Pyridylmethyl N-(2,3-xylyl)anthranilate. USE:An anti-inflammatory and analgesic agent for external use, having high safety, excellent percutaneous absorbability, and capable of exhibiting remarkable anti-inflammatory and analgesic action by application to the affected part. PREPARATION:N-(2,3-Xylyl)anthranilic acid or a halide thereof is reacted with a pyridylalkyl alchol or an alkali N-(2,3-xylyl)anthranilate is reacted with a halide of the pyridylalkyl alcohol to afford the aimed compound expressed by the formula.
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