发明名称 AZAINDOLE DERIVATIVE.
摘要 The purpose of the present invention is to provide a novel compound having a selective JAK3-inhibiting effect and excellent oral absorption. Moreover, the purpose of the present invention is to provide a medical drug useful, on the basis of a JAK3-inhibiting effect, for the prevention and/or treatment of JAK3-associated disease, particularly rheumatoid arthritis or multiple sclerosis. Provided is an azaindole derivative, or a salt thereof, having a cycloalkenyl group that is represented by formula (I) [where R1-R4, m and n are as defined in the Specification], and a medical drug composition comprising the azaindole derivative or salt thereof.
申请公布号 MX2016010078(A) 申请公布日期 2016.10.07
申请号 MX20160010078 申请日期 2015.02.04
申请人 TAIHO PHARMACEUTICAL CO., LTD. 发明人 MITSUYA, Morihiro;NAKAMURA, Masayuki;Hiroyoshi YAMANAKA;Kazuaki SHIBATA;Takafumi HARADA
分类号 C07D471/04;A61K31/437;A61K31/444;A61P1/04;A61P3/10;A61P11/00;A61P11/02;A61P11/06;A61P17/00;A61P17/04;A61P17/06;A61P19/02;A61P21/00;A61P25/00;A61P25/28;A61P27/14;A61P27/16;A61P29/00;A61P31/12;A61P35/00;A61P35/02;A61P37/02;A61P37/06;A61P37/08;A61P43/00 主分类号 C07D471/04
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