ANTIMIGRAINE 4-PYRIMIDINYL AND PYRIDINYL DERIVATIVES OF INDOL-3YL-ALKYL PIPERAZINES
摘要
CT 2148A A series of novel alkoxypyridin-4-yl and alkoxypyrimidin-4-yl derivatives of indol-3-ylalkylpiperazines are intended to be useful agents for alleviation of vascular headache on the basis of their potent affinity and agonist activity at 5-HTID binding sites.
申请公布号
CA2084531(A1)
申请公布日期
1993.06.20
申请号
CA19922084531
申请日期
1992.12.04
申请人
BRISTOL-MYERS SQUIBB COMPANY
发明人
SMITH, DAVID W.;YEVICH, JOSEPH P.;WILLIAMS, ANDREW;RUEDIGER, EDWARD H.;COMBRINK, KEITH D.;PEARCE, BRADLEY C.;YOCCA, FRANK D.;MATTSON, RONALD J.