发明名称 ANTIMIGRAINE 4-PYRIMIDINYL AND PYRIDINYL DERIVATIVES OF INDOL-3YL-ALKYL PIPERAZINES
摘要 CT 2148A A series of novel alkoxypyridin-4-yl and alkoxypyrimidin-4-yl derivatives of indol-3-ylalkylpiperazines are intended to be useful agents for alleviation of vascular headache on the basis of their potent affinity and agonist activity at 5-HTID binding sites.
申请公布号 CA2084531(A1) 申请公布日期 1993.06.20
申请号 CA19922084531 申请日期 1992.12.04
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 SMITH, DAVID W.;YEVICH, JOSEPH P.;WILLIAMS, ANDREW;RUEDIGER, EDWARD H.;COMBRINK, KEITH D.;PEARCE, BRADLEY C.;YOCCA, FRANK D.;MATTSON, RONALD J.
分类号 A61K31/495;A61K31/40;A61K31/44;A61K31/505;A61K31/506;A61P25/04;A61P25/06;C07D209/10;C07D213/65;C07D239/36;C07D241/04;C07D401/12;C07D401/14;C07D403/12;C07D403/14;(IPC1-7):C07D403/14 主分类号 A61K31/495
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