2-SACCHARINYLMETHYL ARYL CARBOXYLATES USEFUL AS PROTEOLYTIC ENZYME INHIBITORS AND COMPOSITIONS AND METHOD OF USE THEREOF
摘要
4-R4-R5-2-Saccharinylmethyl aryl carboxylates, useful in the treatment of degenerative diseases, are prepared by reacting a 4-R4-R5-2-halomethylsaccharin with an arylcarboxylic acid in the presence of an acid-acceptor.
申请公布号
CA2105731(A1)
申请公布日期
1994.04.24
申请号
CA19932105731
申请日期
1993.09.08
申请人
STERLING WINTHROP INC.
发明人
DUNLAP, RICHARD P.;BOAZ, NEIL W.;MURA, ALBERT J.;KUMAR, VIRENDRA;SUBRAMANYAM, CHAKRAPANI;DESAI, RANJIT C.;HLASTA, DENNIS J.;SAINDANE, MANOHAR T.;BELL, MALCOLM R.;COURT, JOHN J.
