发明名称 |
PROCESSES FOR PREPARATION OF EVEROLIMUS AND INTERMEDIATES THEREOF |
摘要 |
The present disclosure discloses processes of Everolimus and intermediates: reacting Sirolimus (Rapamycin) under solvent free conditions with appropriate side chain implying portion wise additions, one pot conversion, and resin mediated synthesis. |
申请公布号 |
CA2818225(C) |
申请公布日期 |
2016.10.25 |
申请号 |
CA20112818225 |
申请日期 |
2011.11.17 |
申请人 |
BIOCON LIMITED |
发明人 |
VENKATA, SRINIVAS PULLELA,;EKAMBARAM, GANESH;KOTHAKONDA, KIRAN KUMAR;PRASAD, ANEGONDI SREENIVASA |
分类号 |
C07D498/18;C07F7/18 |
主分类号 |
C07D498/18 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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