发明名称 4-DIPHENYLACETOXY-N-SUBSTITUTED PIPERIDINES WITH ANTIMUSCARINIC ACTIVITY
摘要 Compounds of formula (I) in which R1 and R2 are each separately selected from a phenyl group which is unsubstituted or substituted by one or more groups selected from alkyl, alkoxy, alkylenedioxy, halogeno, halogeno substituted alkyl, hydroxy and nitro, R3 and R4 are each hydrogen or together are an oxo group and R5 is an alicyclic hydrocarbyl group containing from 3 to 9 carbon atoms in the ring, the compound optionally being in the form of a physiologically acceptable acid addition or quaternary ammonium salt, are of value as selective antagonists of the M3 muscarinic receptor.
申请公布号 AU2673892(A) 申请公布日期 1993.05.03
申请号 AU19920026738 申请日期 1992.10.08
申请人 BRITISH TECHNOLOGY GROUP LTD 发明人 RICHARD BAWDEN BARLOW;MARK ANTHONY VEALE
分类号 C07D211/46 主分类号 C07D211/46
代理机构 代理人
主权项
地址